From Wikipedia, the free encyclopedia
Chemical compound
Fazadinium bromide is a
muscle relaxant which acts as a
nicotinic acetylcholine receptor
antagonist through
neuromuscular blockade.
[1]
References
-
^ Camu F, D'Hollander A (1978). "Neuromuscular blockade of fazadinium bromide (AH 8165) in renal failure patients". Acta Anaesthesiologica Scandinavica. 22 (3): 221–6.
doi:
10.1111/aas.1978.22.3.221.
PMID
27936.
|
---|
nAChRsTooltip Nicotinic acetylcholine receptors |
Agonists (and
PAMsTooltip positive allosteric modulators) |
-
5-HIAA
-
6-Chloronicotine
-
A-84,543
-
A-366,833
-
A-582,941
-
A-867,744
-
ABT-202
-
ABT-418
-
ABT-560
-
ABT-894
-
Acetylcholine
-
Altinicline
-
Anabasine
-
Anatabine
-
Anatoxin-a
-
AR-R17779
-
Bephenium hydroxynaphthoate
-
Butinoline
-
Butyrylcholine
-
Carbachol
-
Choline
-
Cotinine
-
Cytisine
-
Decamethonium
-
Desformylflustrabromine
-
Dianicline
-
Dimethylphenylpiperazinium
-
Epibatidine
-
Epiboxidine
-
Ethanol (alcohol)
-
Ethoxysebacylcholine
-
EVP-4473
-
EVP-6124
-
Galantamine
-
GTS-21
-
Ispronicline
-
Ivermectin
-
JNJ-39393406
-
Levamisole
-
Lobeline
-
MEM-63,908 (RG-3487)
-
Morantel
-
Nicotine (
tobacco)
-
NS-1738
-
PHA-543,613
-
PHA-709,829
-
PNU-120,596
-
PNU-282,987
-
Pozanicline
-
Pyrantel
-
Rivanicline
-
RJR-2429
-
Sazetidine A
-
SB-206553
-
Sebacylcholine
-
SIB-1508Y
-
SIB-1553A
-
SSR-180,711
-
Suberyldicholine
-
Suxamethonium (succinylcholine)
-
Suxethonium (succinyldicholine)
-
TC-1698
-
TC-1734
-
TC-1827
-
TC-2216
-
TC-5214
-
TC-5619
-
TC-6683
-
Tebanicline
-
Tribendimidine
-
Tropisetron
-
UB-165
-
Varenicline
-
WAY-317,538
-
XY-4083
|
---|
Antagonists (and
NAMsTooltip negative allosteric modulators) | |
---|
|
---|
Precursors (and
prodrugs) | |
---|
|